Saxsons Group
Lu-177 n.c.a. lutetium chloride solution in shielded transport vial
≥3,000 GBq/mg
specific activity
≥99.9 %
radionuclidic purity
6.647 day
half-life
n.c.a.
no carrier added
37 GBq/mL
activity concentration

Authorised Indian Distributor

Saxsons Group

New Delhi, India · Since 1997

SX
Nuclear Medicine NM-017 AERB Importable No-Carrier-Added cGMP · ICH-Q7 FDA DMF supported

Lu-177 n.c.a. No-Carrier-Added Lutetium-177 — Theranostic Building Block

The starting material for every Lu-177 theranostic protocol — produced by SHINE Medical in Janesville, Wisconsin and supplied across India by Saxsons. No-carrier-added ¹⁷⁷LuCl₃ in 0.04 M HCl, ≥99.9 % radionuclidic purity, ≥3,000 GBq/mg specific activity at calibration. The chemistry inputs that decide PSMA-617, DOTATATE and FAPI labelling yields. Cold-chain delivered across India with AERB import documentation.

Key Features

  • No-carrier-added (n.c.a.) production — no stable Lu-176 / Lu-175 carrier in the matrix, the highest specific activity reachable in clinical supply
  • Specific activity ≥3,000 GBq/mg at calibration, with batches reaching ≈3,700 GBq/mg — the same Lu-177 mass carries far more radioactive atoms, so the labelling kit competes against fewer cold lutetium ions
  • Radionuclidic purity ≥99.9 % ¹⁷⁷Lu at calibration (Ph. Eur. compliant)
  • Lu-177m metastable contamination held to negligible levels — the long-lived 160-day isomer that drives carrier-added waste decisions is essentially absent, so spent-vial waste decays on the ~6.65-day primary half-life
  • Standard chemical form: ¹⁷⁷LuCl₃ in 0.04 M HCl — drop-in compatible with PSMA-617, DOTATATE, FAPI-46 and DOTA-conjugate radiolabelling SOPs
View all features

All Features

  • No-carrier-added (n.c.a.) production — no stable Lu-176 / Lu-175 carrier in the matrix, the highest specific activity reachable in clinical supply
  • Specific activity ≥3,000 GBq/mg at calibration, with batches reaching ≈3,700 GBq/mg — the same Lu-177 mass carries far more radioactive atoms, so the labelling kit competes against fewer cold lutetium ions
  • Radionuclidic purity ≥99.9 % ¹⁷⁷Lu at calibration (Ph. Eur. compliant)
  • Lu-177m metastable contamination held to negligible levels — the long-lived 160-day isomer that drives carrier-added waste decisions is essentially absent, so spent-vial waste decays on the ~6.65-day primary half-life
  • Standard chemical form: ¹⁷⁷LuCl₃ in 0.04 M HCl — drop-in compatible with PSMA-617, DOTATATE, FAPI-46 and DOTA-conjugate radiolabelling SOPs
  • Standard activity concentration 1.0 Ci/mL (37 GBq/mL) at calibration
  • Produced by SHINE Medical (Janesville, Wisconsin) under cGMP and ICH-Q7; supported by an FDA Drug Master File
  • Cold-chain delivery from production to Indian hospital pharmacy — calibration to a defined date/time so the dose lands ready for labelling on therapy day
  • AERB sealed / unsealed source import documentation handled by Saxsons
  • Certificate of Analysis, radionuclidic purity report and batch release documentation with every shipment
  • Compatible with ¹⁷⁷Lu-DOTATATE PRRT, ¹⁷⁷Lu-PSMA-617 prostate theranostics and ¹⁷⁷Lu-FAPI emerging-tumour-stroma protocols — the same starting material across all three
  • Dosimetry consultation available for cycle planning (208 keV imaging gamma for post-therapy SPECT/CT)

Technical Specifications

Radionuclide Lutetium-177 (¹⁷⁷Lu)
Production route No-carrier-added (n.c.a.) — no stable Lu carrier in the matrix
Half-life 6.647 days
Decay mode β⁻ (Eβ,max 498 keV; mean 134 keV) + γ 113 keV (6.4 %), 208 keV (11 %)
Specific activity ≥3,000 GBq/mg at calibration; batch peaks ≈3,700 GBq/mg
Activity concentration 1.0 Ci/mL (37 GBq/mL) at standard calibration time
Chemical form n.c.a. ¹⁷⁷LuCl₃ in 0.04 M HCl solution
Radionuclidic purity ≥99.9 % ¹⁷⁷Lu (Ph. Eur. compliant)
Radiochemical purity ≥99 % as ¹⁷⁷LuCl₃
Lu-177m contamination Negligible — long-lived (≈160 d) isomer effectively absent; waste decays on ≈6.65 d half-life
Manufacturer SHINE Medical Technologies (Janesville, Wisconsin, USA)
Regulatory framework cGMP, ICH-Q7, FDA-21CFR; supported by SHINE FDA Drug Master File
Labelling compatibility PSMA-617 · DOTATATE · FAPI-46 · DOTA-conjugate peptides
AERB status Import licence required; Saxsons manages regulatory documentation

Applications

One n.c.a. Lu-177 supply chain — DOTATATE, PSMA, FAPI and beyond

¹⁷⁷Lu-DOTATATE PRRT

Peptide receptor radionuclide therapy in somatostatin-receptor-positive gastroenteropancreatic and bronchopulmonary NETs. n.c.a. purity maximises peptide labelling yield and minimises cold-DOTATATE competition for SSTR2 binding sites.

¹⁷⁷Lu-PSMA-617 mCRPC therapy

Targeted β-radiation to PSMA-expressing prostate cancer cells in metastatic castration-resistant disease. n.c.a. delivers the high specific activity required for dosimetry-guided multi-cycle planning.

¹⁷⁷Lu-FAPI tumour-stroma

Emerging fibroblast-activation-protein-targeted therapy across pancreatic, sarcoma, breast and other FAP-positive tumours. n.c.a. Lu-177 is the regulatory-compliant starting material for clinical and academic FAPI protocols.

Theranostic pairing with Ga-68 PET

Same molecular target on the diagnostic and therapeutic side — Ga-68 DOTATATE / PSMA / FAPI on PET, ¹⁷⁷Lu on therapy. n.c.a. Lu-177 keeps the imaging-therapy chain consistent on specific activity.

Post-therapy SPECT/CT dosimetry

The 208 keV gamma emission enables quantitative SPECT/CT imaging after each Lu-177 cycle. n.c.a. activity per peptide lets the dosimetrist resolve tumour and organ uptake at clinical activity levels.

Investigator-initiated trials

Academic theranostic programmes in India (AIIMS, Tata Memorial, BARC-collaborating centres) use n.c.a. Lu-177 for novel-peptide protocols. Saxsons supports IND-equivalent documentation and audit trail.

Why Lu-177 n.c.a.?

≥3,000 GBq/mg
Specific activity that the kit can see

A labelling kit competes for binding sites against any cold lutetium in the matrix. Carrier-added Lu-177 typically lands at ~600 GBq/mg; n.c.a. at ≥3,000 GBq/mg means roughly 5× fewer cold-Lu atoms per labelled molecule. That difference shows up directly as higher labelling yield, lower DOTATATE / PSMA-617 / FAPI dose, and a cleaner tumour-to-background ratio at imaging.

Negligible ¹⁷⁷ᵐLu
Waste decays in days, not months

Carrier-added Lu-177 carries a Lu-177m (metastable, T½ ≈160 d) impurity. That contaminant drives long-tail kidney dose during therapy and a long decay-store dwell time for vials and patient excreta. n.c.a. production effectively eliminates Lu-177m, so the spent-vial waste decays on the primary 6.65-day half-life — practical decay-store rotation, lower cumulative organ dose.

cGMP + FDA DMF
Regulatory dossier already built

SHINE Medical produces the starting material under cGMP and ICH-Q7, with an FDA Drug Master File on file. For an Indian centre running DOTATATE, PSMA or FAPI under AERB licensing or hospital ethics-committee oversight, the upstream regulatory dossier is already assembled — Saxsons supplies the import-side licensing paperwork from there.

Catalogs & Resources

SHINE product page. Contact Saxsons for AERB import documentation, calibration date scheduling and India pricing.

Available through Saxsons Group

Build your Lu-177 theranostic supply chain on n.c.a. starting material

Contact Saxsons Group for n.c.a. Lu-177 supply agreements, AERB import documentation and cold-chain scheduling across India — for DOTATATE, PSMA-617 and FAPI programmes alike.